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Frontiers | A Review of the Therapeutic Potential of Recently Developed G  Protein-Biased Kappa Agonists
Frontiers | A Review of the Therapeutic Potential of Recently Developed G Protein-Biased Kappa Agonists

The Role of Dynorphin and the Kappa Opioid Receptor in the Symptomatology  of Schizophrenia: A Review of the Evidence
The Role of Dynorphin and the Kappa Opioid Receptor in the Symptomatology of Schizophrenia: A Review of the Evidence

Elucidating the active δ-opioid receptor crystal structure with peptide and  small-molecule agonists | Science Advances
Elucidating the active δ-opioid receptor crystal structure with peptide and small-molecule agonists | Science Advances

Nanobody-enabled monitoring of kappa opioid receptor states | Nature  Communications
Nanobody-enabled monitoring of kappa opioid receptor states | Nature Communications

Table 1 from Discovery of the First Small-Molecule Opioid Pan Antagonist  with Nanomolar Affinity at Mu, Delta, Kappa, and Nociceptin Opioid  Receptors | Semantic Scholar
Table 1 from Discovery of the First Small-Molecule Opioid Pan Antagonist with Nanomolar Affinity at Mu, Delta, Kappa, and Nociceptin Opioid Receptors | Semantic Scholar

A Narrative Pharmacological Review of Buprenorphine: A Unique Opioid for  the Treatment of Chronic Pain | Pain and Therapy
A Narrative Pharmacological Review of Buprenorphine: A Unique Opioid for the Treatment of Chronic Pain | Pain and Therapy

Kappa opioid receptor binding affinity and the effects on... | Download  Scientific Diagram
Kappa opioid receptor binding affinity and the effects on... | Download Scientific Diagram

Structure-Based Discovery of New Antagonist and Biased Agonist Chemotypes  for the Kappa Opioid Receptor | Journal of Medicinal Chemistry
Structure-Based Discovery of New Antagonist and Biased Agonist Chemotypes for the Kappa Opioid Receptor | Journal of Medicinal Chemistry

Antagonists of the kappa opioid receptor - ScienceDirect
Antagonists of the kappa opioid receptor - ScienceDirect

Novel Mixed NOP/Opioid Receptor Peptide Agonists | Journal of Medicinal  Chemistry
Novel Mixed NOP/Opioid Receptor Peptide Agonists | Journal of Medicinal Chemistry

Molecular mechanism of biased signaling at the kappa opioid receptor |  Nature Communications
Molecular mechanism of biased signaling at the kappa opioid receptor | Nature Communications

Frontiers | A Review of the Therapeutic Potential of Recently Developed G  Protein-Biased Kappa Agonists
Frontiers | A Review of the Therapeutic Potential of Recently Developed G Protein-Biased Kappa Agonists

Chemical structures of 'affinity-dominant' and 'efficacy-dominant' G... |  Download Scientific Diagram
Chemical structures of 'affinity-dominant' and 'efficacy-dominant' G... | Download Scientific Diagram

Molecules | Free Full-Text | Ligand-Free Signaling of G-Protein-Coupled  Receptors: Relevance to μ Opioid Receptors in Analgesia and Addiction
Molecules | Free Full-Text | Ligand-Free Signaling of G-Protein-Coupled Receptors: Relevance to μ Opioid Receptors in Analgesia and Addiction

Kappa Opiate Receptor Agonist - an overview | ScienceDirect Topics
Kappa Opiate Receptor Agonist - an overview | ScienceDirect Topics

PDF] The Roles of Opioid Receptors and Agonists in Health and Disease  Conditions | Semantic Scholar
PDF] The Roles of Opioid Receptors and Agonists in Health and Disease Conditions | Semantic Scholar

Pharmaceuticals | Free Full-Text | Biased, Bitopic, Opioid–Adrenergic  Tethered Compounds May Improve Specificity, Lower Dosage and Enhance Agonist  or Antagonist Function with Reduced Risk of Tolerance and Addiction
Pharmaceuticals | Free Full-Text | Biased, Bitopic, Opioid–Adrenergic Tethered Compounds May Improve Specificity, Lower Dosage and Enhance Agonist or Antagonist Function with Reduced Risk of Tolerance and Addiction

Human native kappa opioid receptor functions not predicted by recombinant  receptors: Implications for drug design | Scientific Reports
Human native kappa opioid receptor functions not predicted by recombinant receptors: Implications for drug design | Scientific Reports

κ-opioid receptor - Wikipedia
κ-opioid receptor - Wikipedia

Molecules | Free Full-Text | Design of κ-Opioid Receptor Agonists for  the Development of Potential Treatments of Pain with Reduced Side Effects
Molecules | Free Full-Text | Design of κ-Opioid Receptor Agonists for the Development of Potential Treatments of Pain with Reduced Side Effects

Opioid Receptor Binding Affinities of Dynorphin Analogues. | Download Table
Opioid Receptor Binding Affinities of Dynorphin Analogues. | Download Table

Noribogaine is a G-protein biased κ-opioid receptor agonist - ScienceDirect
Noribogaine is a G-protein biased κ-opioid receptor agonist - ScienceDirect

Binding affinity, potency, and intrinsic activity of opioid ligands in... |  Download Table
Binding affinity, potency, and intrinsic activity of opioid ligands in... | Download Table

Opioid receptors | Introduction | BPS/IUPHAR Guide to PHARMACOLOGY
Opioid receptors | Introduction | BPS/IUPHAR Guide to PHARMACOLOGY